Enzyme inhibitors
| Catalog | Product Name / CAS / Description | Structure |
|---|---|---|
| BBF-03109 |
Tetrafibricin (151705-56-5) Inquiry |
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Tetrafibricin is a fibrinogen antagonist produced by Str. neyagawaensis NR0577. Tetrafibricin has a strong inhibitory effect on the binding of fibrinogen to the GP IIb/IIIa receptor with an IC50 of 46 nmol/L, and an IC50 of 46 mol/L for the inhibition of HeLa cell toxicity. |
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| BBF-03117 |
Tetronothiodin (139643-79-1) Inquiry |
|
Tetronothiodin is a trypsin secretin type B receptor antagonist produced by Str. sp. NR0489. Tetronothiodin can inhibit the binding of trypsin C-terminal 8 peptide to rat cortical trypsin B receptor, with IC50 of 3.6 µmol/L. |
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| BBF-03124 | ||
Thielavin D is a glucose-6-phosphatase (G6Pase) inhibitor produced by Chaetomium carinthiacum. |
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| BBF-03125 | ||
Thielavin P is a glucose-6-phosphatase (G6Pase) inhibitor produced by Chaetomium carinthiacum. |
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| BBF-03161 | ||
A58365 A is an enzyme inhibitor produced by Streptomyces chromofuscus A58365.1. It has the effect of inhibiting angiotensin transferase (ACE). |
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| BBF-03162 | ||
A58365 B is an enzyme inhibitor produced by Streptomyces chromofuscus A58365.1. It has the effect of inhibiting angiotensin transferase (ACE). |
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| BBF-03163 | ||
A-72363 A1 is a Heparanase inhibitor produced by Streptomyces nobilis SANK 60192. |
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| BBF-03164 | ||
A-72363 A2 is a Heparanase inhibitor produced by Streptomyces nobilis SANK 60192. |
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| BBF-03165 | ||
A-72363 C is a Heparanase inhibitor produced by Streptomyces nobilis SANK 60192. |
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| BBF-03166 | ||
A-75943 is is a bone resorption inhibitor produced by Streptomyces sp. SANK61296. In vitro tests, it has the effect of inhibiting bone resorption with IC50 of 0.35 µmol/L. It also inhibits the bone resorption in rats with thyroid and parathyroidectomy. |
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| BBF-03205 | ||
AM 4299 A is a thiol protease inhibitor produced by Chromelosporium fulvum M4299. |
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| BBF-03206 | ||
AM 4299 B is a thiol protease inhibitor produced by Chromelosporium fulvum M4299. |
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| BBF-03207 | ||
AS-183 is an enzyme inhibitor produced by Scedosporium sp. SPC-15549. |
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| BBF-03208 |
Penicillide (55303-92-9) Inquiry |
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Penicillide is an acyl-CoA: cholesterol acyltransferase (ACAT) inhibitor produced by Penicillum asperosporum KY1635. The IC50 for inhibiting ACAT was 22.9 µmol/L. |
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| BBF-03209 | ||
AS-186c is an acyl-CoA: cholesterol acyltransferase (ACAT) inhibitor produced by Penicillum asperosporum KY1635. The IC50 for inhibiting ACAT was 11.5 µmol/L. |
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| BBF-03210 | ||
AS-186d is an acyl-CoA: cholesterol acyltransferase (ACAT) inhibitor produced by Penicillum asperosporum KY1635. The IC50 for inhibiting ACAT was 12.4 µmol/L. |
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| BBF-03216 |
Mer-NF5003F (149598-70-9) Inquiry |
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Mer-NF5003F is a myo-inositol monophosphatase (IMPase) inhibitor produced by Memnoniella echinata. |
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| BBF-03217 | ||
L-671776 is a myo-inositol monophosphatase (IMPase) inhibitor produced by Memnoniella echinata. |
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| BBF-03218 |
Mer-NF5003E (159121-98-9) Inquiry |
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Mer-NF5003E is a myo-inositol monophosphatase (IMPase) inhibitor produced by Memnoniella echinata. |
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| BBF-03219 | ||
B-5354a is a Sphingosine kinase (SPHK) inhibitor produced by SANK 71896. It has the activity of inhibiting SPHK with IC50 of 21 µmol/L. |
